Compound Reference Overview
| Field | Value |
|---|---|
| Name | NA-Selank (N-Acetyl Selank) |
| Reference Code | SELANK |
| Category | Cognitive / Anxiolytic Peptide |
| Example Strength | 10 mg vial (varies by manufacturer) |
| Reference Range | 250–1000 mcg once daily |
| Frequency | Once daily |
| Key Safety Warning | Not FDA-approved. Limited large-scale human trials outside Russia. Use caution when combined with other anxiolytics. |
Mechanism of Action (Educational)
NA-Selank is an N-acetylated synthetic analog of Selank, a heptapeptide derived from tuftsin. It modulates GABAergic signaling and influences serotonin and dopamine pathways.
Research suggests Selank may enhance brain-derived neurotrophic factor (BDNF) expression and regulate cytokine activity, contributing to anxiolytic and cognitive-enhancing effects without significant sedation.
Indications (Literature / Off-Label)
- Anxiety and stress modulation
- Cognitive enhancement
- Learning and memory support
- Stress-related cognitive impairment
Administration (Literature)
| Parameter | Details |
|---|---|
| Route | Subcutaneous or intranasal |
| Frequency | Once daily |
| Injection Sites | Subcutaneous: abdomen Intranasal: divided between nostrils |
| Timing | Morning or as needed for anxiety; adjust based on fatigue response |
Titration Schedule (Literature)
- Weeks 1–2: 250–500 mcg once daily
- Weeks 3+: 500–750 mcg daily based on response
- Maximum commonly referenced range: 1000 mcg daily
Adjust timing if fatigue occurs.
Pharmacokinetics (Literature)
- Rapid CNS activity observed (minutes to hours)
- Anxiolytic effects reported within hours to days
- Human pharmacokinetic data remain limited
Reconstitution & Concentration
(Mathematical Illustration Only)
| Parameter | Value |
|---|---|
| Diluent | Bacteriostatic water (example only) |
| Reconstitution Volume | 2 mL (example) |
| Resulting Concentration | 5 mg/mL (5000 mcg/mL) |
| Stability | Up to 28 days refrigerated (varies by formulation) |
Reconstitution Math Example
- 10 mg ÷ 2 mL = 5 mg/mL
- 0.1 mL = 500 mcg
- 0.2 mL = 1000 mcg
Provided strictly for arithmetic reference.
Mathematical Calculation Tool
The calculator below allows concentration and volume calculations based on vial strength and dilution volume. This tool is provided strictly for mathematical reference.
Peptide Reconstitution Calculator
For Educational & Professional Reference Only
Safety & Contraindications (Summary)
Contraindications
- Pregnancy or breastfeeding
- Known hypersensitivity
Drug Interactions
- Benzodiazepines (moderate): additive anxiolytic effect
Adverse Events
- Fatigue
- Nasal irritation (intranasal use)
- Headache
Serious Risks
- Rare in available literature
Monitoring (Literature)
- Anxiety levels
- Mood changes
- Cognitive performance
Disclaimer
NA-Selank is not FDA-approved. This content is provided strictly for educational and professional reference purposes. All clinical decisions must be made by a licensed healthcare professional.
Reference Sources
1. Zozulya AA, et al. Effects of Selank on GABAergic neurotransmission.
Bull Exp Biol Med. 2003.
2. Volkova AV, et al. Selank effects on BDNF expression and anxiety models.
Neurosci Behav Physiol. 2011.
3. Andreeva LA, et al. Clinical use of Selank in anxiety disorders.
Zh Nevrol Psikhiatr Im S S Korsakova. 2005.